Comparison of the cytotoxic effects of enantiopure PPAPs, including nemorosone and clusianone.

نویسندگان

  • Nigel S Simpkins
  • Frank Holtrup
  • Vincent Rodeschini
  • James D Taylor
  • Robert Wolf
چکیده

The synthesis of an unnatural polyprenylated acylphloroglucinol (PPAP), regioisomeric with nemorosone and clusianone, has been accomplished. The separated enantiomers of this new PPAP, along with those of nemorosone and clusianone, have been screened for activity against HeLa (cervix carcinoma), MIA-PaCa-2 (pancreatic carcinoma), and MCF7 (mamma carcinoma) cancer cell lines. All of the isomers examined gave surprisingly similar results in the screens.

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عنوان ژورنال:
  • Bioorganic & medicinal chemistry letters

دوره 22 19  شماره 

صفحات  -

تاریخ انتشار 2012